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  • 產(chǎn)品名稱: EZM0414
  • 產(chǎn)品貨號(hào): CST9969
  • 貨期: 現(xiàn)貨
  • 價(jià)格與訂購(gòu): 2800
  • 數(shù)量:
    庫(kù)存: 5
  • 規(guī)格: 1mg
  • 產(chǎn)品信息
  • 如何訂購(gòu)
    產(chǎn)品描述
    EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay. EZM0414 can be used for the research of relapsed or refractory multiple myeloma and diffuse large B-cell lymphoma [1].
    Cas No.
    2411748-50-8
    分子式
    C22H29FN4O2
    分子量
    400.49
    參考文獻(xiàn)
    [1]Jennifer Totman, et al. Pharmacologic Inhibition of the Histone Methyltransferase SETD2 with EZM0414 As a Novel Therapeutic Strategy in Relapsed or Refractory Multiple Myeloma and Diffuse Large B-cell Lymphoma.
    儲(chǔ)存和溶解度
    DMSO:115 mg/mL (287.15 mM),ultrasonic and warming and heat to 60°C
    Powder: -20°C for 3 years
    In solvent: -80°C for 2 years
    Note
    For research use only .
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